erk2 in-1 — TargetMol Chemicals

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Search Results for " erk2 in-1 "

Compounds

Cat No.	Product Name	Synonyms	Targets
T11228	ERK2 IN-1		ERK
	ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM.		ERK
T2310L	CHIR-99021 HCl	CT99021 HCl,Laduviglusib HCl	GSK-3
	CHIR-99021 HCl (Laduviglusib HCl) is a highly potent and selective inhibitor of GSK-3α/β, with IC50 values of 10 nM and 6.7 nM respectively. It demonstrates remarkable selectivity for GSK-3, with over 500-fold selectivit...		GSK-3
T6S0655	Corynoxeine		ERK
	1. Corynoxeine is a potent ERK1/2 inhibitor of key PDGF-BB-induced VSMC proliferation and may be useful in the prevention and treatment of vascular diseases and restenosis after angioplasty.		ERK
T76556	MEK1 Derived Peptide Inhibitor 1
	MEK1 Derived Peptide Inhibitor 1, a peptide inhibitor, prevents the in vitro activation of ERK2 by MEK1, exhibiting an inhibitory concentration (IC 50) of 30 μM. It is utilized in the study of cell-permeable [1].
T11225	ERK-IN-2		ERK
	ERK-IN-2, an ERK2 inhibitor, exhibits an IC50 value of 1.8 nM. At doses greater than 10 μM, it may induce off-target toxicity and/or activity [1].		ERK
T81387	Prosaptide Tx14(A) TFA
	Prosaptide Tx14(A) TFA is a prosaposin-derived peptide and a potent agonist of both GPR37L1 and GPR37, exhibiting EC50 values of 5 nM and 7 nM, respectively. In Schwann cells, this compound enhances phosphorylation of bo...
T61755	E6201
	E6201 (ER-806201) is a potent dual kinase inhibitor targeting MEK1 and FLT3, inhibiting their activities in an ATP-competitive manner. It effectively suppresses MEK1-induced ERK2 phosphorylation (IC50 = 5.2 nM), MKK4-ind...
T38377	ADTL-EI1712	ADTL-EI1712
	ADTL-EI1712 is a dual inhibitor of ERK1 and ERK5 (IC50s = 40.43 and 64.5 nM, respectively).1It reduces ERK1 and ERK5 activity by 93.5% and 89.4%, respectively, but also inhibits ERK2 activity by 92.7%, in a panel of 100 ...